ShK-Dap22 TFA is a potent and specific Kv1.3 immunosuppressive polypeptide. It acts as a selective Kv1.3 channel blocker, exhibiting IC50 values of 23 pM for mKv1.3, 1.8 nM for mKv1.1, 10.5 nM for hKv1.6, 37 nM for mKv1.4, and 39 nM for rKv1.2 channels.
Formel:
C168H269F3N54O50S7
Target-Kategorie:
Others
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