UNC0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases G9a and GLP (IC50s: 6 nM/15 nM for G9a/GLP). UNC0646(UNC 0646) potently blocks G9a/GLP methyltransferase activity in cells (IC50: 10 nM in MCF7 cells) and exhibits low cellular toxicity (EC50: 4.7 µM in MCF7 cells).
Molekulargewicht:
621.9
Reinheit:
>99.99%
CAS Nummer:
[1320288-17-2]
Formel:
C36H59N7O2
Target-Kategorie:
Histone Methyltransferase
TQ0232
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