A synthetic agonist of the cannabinoid receptor 1 (CB1R). ACEA is considered to be a selective cannabinoid agonist as it binds primarily to the CB1R and has low affinity to the cannabinoid receptor 2 (CB2R). A potent and highly selective agonist for CB1 receptor. Affinity for CB1 (Ki = 1.4nM) is more than1400-fold higher than that for CB2 (KMGK = 3100nM) receptors. Synonyms: (5Z,8Z,11Z,14Z)-N-(2-Chloroethyl)-5,8,11,14-eicosatetraenamide, ACEA, 2-chloro-AEA CAS No: 220556-69-4 Molecular Formula: C22H36ClNO Molecular Weight: 365.99 Purity: 95% (HPLC) Appearance: Solution in methyl acetate Solubility: Soluble in Ethanol, DMSO, and DMF Infared Radiation: Conforms to structure Method for Determining Identity: Mass Spectometry Primary Target: CB1 receptor Primary Target Ki: 1.4nM and 3100nM for CB1 and CB2 receptors, respectively. Storage and Stability: Aliquot to avoid repeated freezing and thawing and store at -70C. Aliquots are stable for 6 months after receipt. For maximum recovery of product, centrifuge the original vial after thawing and prior to removing the cap.
Molekulargewicht:
365.99
CAS Nummer:
[220556-69-4]
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