YM298198 Hydrochloride (6-Amino-N-cyclohexyl-N,3-dimethylthiazolo[3,2-a]benzimidazole-2-carboxamide Hydrochloride), CAS [[748758-45-4]]

Artikelnummer: USB-217880
Artikelname: YM298198 Hydrochloride (6-Amino-N-cyclohexyl-N,3-dimethylthiazolo[3,2-a]benzimidazole-2-carboxamide Hydrochloride), CAS [[748758-45-4]]
Artikelnummer: USB-217880
Hersteller Artikelnummer: 217880
Alternativnummer: USB-217880-10
Hersteller: US Biological
Kategorie: Biochemikalien
A highly potent antagonist selective for mGlu1 receptors (IC50 = 16nM). Biologically active admitted orally or systematically. Often used in assessing the functional roles of mGlu1 receptors in a variety of research areas, such as anxiety and stress related disorders, analgesia, nociceptive pain, and schizophrenia. CAS Number: 748758-45-4 Formula: C18H22N4OSHCl Solubility: H2O Primary Target: mGlu1 receptors Primary Target IC50: 16nM Storage and Stability: May be stored at 4C. For long-term storage, aliquot and store at 4C. Do not freeze. For maximum recovery of product, centrifuge the original vial prior to removing the cap. Further dilutions can be made in assay buffer.
Reinheit: 99% (HPLC)
Formulierung: Supplied as a cream solid.
CAS Nummer: [748758-45-4]