2-APB, CAS [[524-95-8]]

Artikelnummer: USB-254353
Artikelname: 2-APB, CAS [[524-95-8]]
Artikelnummer: USB-254353
Hersteller Artikelnummer: 254353
Alternativnummer: USB-254353-10, USB-254353-50
Hersteller: US Biological
Kategorie: Biochemikalien
A functional and membrane permeable D-myo-inositol 1,4,5-trisphosphate (IP3) receptor antagonist (IC50 = 42uM). Stimulates store-operated calcium (SOC) release at low concentrations (< 10uM) and inhibits it at higher concentrations (up to 50uM). Increases STIM-Orai channel conductance and limits ion selectivity. Modulator of TRP channels, blocks TRPC1, TRPC3, TRPC5, TRPC6, TRPV6, TRPM3, TRPM7, TRPM8 and TRPP2 and at higher concentrations stimulates TRPV1, TRPV2 and TRPV3. Also blocks specific gap channel subtypes. CAS Number: 524-95-8
Reinheit: 98%
CAS Nummer: [524-95-8]