GSK5182, CAS [[877387-37-6]]

Produktübersicht

• Artikelname: GSK5182, CAS [[877387-37-6]]
• Artikelnummer: AMO-M20777
• Hersteller Artikelnummer: M20777
• Alternativnummer: AMO-M20777-5MG,AMO-M20777-10MG,AMO-M20777-25MG,AMO-M20777-50MG
• Hersteller: Abmole Bioscience
• Kategorie: Biochemikalien

Produktbeschreibung

GSK5182 is a 4-Hydroxytamoxifen analog and a highly potent, selective, orally active estrogen-related receptor gamma (ERRgamma) inverse agonist with an IC50 value of 79 nM.GSK5182 does not interact with other nuclear receptors, including ERRalpha and ERalpha. In addition, GSK5182 inhibits proinflammatory cytokine-induced catabolic factors and increases ROS production in liver cancer cells. cytokine-induced catabolic factors and increased ROS production in hepatocellular carcinoma cells.

Produkteigenschaften

• Molekulargewicht: 417.54
• Reinheit: >99%
• CAS Nummer: [877387-37-6]
• Formel: C27H31NO3
• Target-Kategorie: Estrogen Receptor