Larotrectinib (LOXO-101), CAS [[1223403-58-4]]

Artikelnummer: AMO-M6151
Artikelname: Larotrectinib (LOXO-101), CAS [[1223403-58-4]]
Artikelnummer: AMO-M6151
Hersteller Artikelnummer: M6151
Alternativnummer: AMO-M6151-2MG,AMO-M6151-5MG,AMO-M6151-10MG,AMO-M6151-50MG
Hersteller: Abmole Bioscience
Kategorie: Biochemikalien
Alternative Synonym: ARRY-470, larotrectinib
Larotrectinib (LOXO-101) is a potent, ATP competitive TRK inhibitor with IC50s in low nanomolar range for inhibition of all TRK family members in binding and cellular assays, with 100x selectivity over other kinases, with 2 to 20 nM cellular potency against the TRKA, TRKB, and TRKC kinases.
Molekulargewicht: 428.44
Reinheit: 99.56%
CAS Nummer: [1223403-58-4]
Formel: C21H22F2N6O2
Target-Kategorie: Trk