Larotrectinib (LOXO-101), CAS [[1223403-58-4]]
Artikelnummer:
AMO-M6151
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| Artikelname: | Larotrectinib (LOXO-101), CAS [[1223403-58-4]] |
| Artikelnummer: | AMO-M6151 |
| Hersteller Artikelnummer: | M6151 |
| Alternativnummer: | AMO-M6151-2MG,AMO-M6151-5MG,AMO-M6151-10MG,AMO-M6151-50MG |
| Hersteller: | Abmole Bioscience |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | ARRY-470, larotrectinib |
| Larotrectinib (LOXO-101) is a potent, ATP competitive TRK inhibitor with IC50s in low nanomolar range for inhibition of all TRK family members in binding and cellular assays, with 100x selectivity over other kinases, with 2 to 20 nM cellular potency against the TRKA, TRKB, and TRKC kinases. |
| Molekulargewicht: | 428.44 |
| Reinheit: | 99.56% |
| CAS Nummer: | [1223403-58-4] |
| Formel: | C21H22F2N6O2 |
| Target-Kategorie: | Trk |
