Varenicline hydrochloride, CAS [[230615-23-3]]
Artikelnummer:
AMO-M9058
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| Artikelname: | Varenicline hydrochloride, CAS [[230615-23-3]] |
| Artikelnummer: | AMO-M9058 |
| Hersteller Artikelnummer: | M9058 |
| Alternativnummer: | AMO-M9058-5MG,AMO-M9058-10MG,AMO-M9058-50MG |
| Hersteller: | Abmole Bioscience |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | CP 526555 hcl, Chantix, Champix |
| Varenicline hydrochloride is a potent partial agonist of alpha4beta2 nicotinic acetylcholine receptor (nAChR) and alpha3beta4 nAChR, with EC50s of 2.3 µM and 55 µM, respectively. In addition, Varenicline hydrochloride is also a potent full agonist of alpha7 nAChRs. In addition, Varenicline hydrochloride is a potent full alpha7 nAChRs agonist with an EC50 of 18 µM. |
| Molekulargewicht: | 247.72 |
| Reinheit: | >98.5% |
| CAS Nummer: | [230615-23-3] |
| Formel: | C13H14ClN3 |
| Target-Kategorie: | AChR/AChE |
