Varenicline hydrochloride is a potent partial agonist of alpha4beta2 nicotinic acetylcholine receptor (nAChR) and alpha3beta4 nAChR, with EC50s of 2.3 µM and 55 µM, respectively. In addition, Varenicline hydrochloride is also a potent full agonist of alpha7 nAChRs. In addition, Varenicline hydrochloride is a potent full alpha7 nAChRs agonist with an EC50 of 18 µM.
Molecular Weight:
247.72
Purity:
>98.5%
CAS Number:
[230615-23-3]
Formula:
C13H14ClN3
Target:
AChR/AChE
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