TZ9, Rad6 Ubiquitin Inhibitor, CAS [[1002789-86-7]], Unconjugated

Artikelnummer: BSS-BS-60286C
Artikelname: TZ9, Rad6 Ubiquitin Inhibitor, CAS [[1002789-86-7]], Unconjugated
Artikelnummer: BSS-BS-60286C
Hersteller Artikelnummer: bs-60286C
Alternativnummer: BSS-BS-60286C-10,BSS-BS-60286C-2
Hersteller: Bioss
Kategorie: Biochemikalien
Konjugation: Unconjugated
TZ9 is a selective and cell permeable inhibitor of human E2 ubiquitin-conjugating enzyme Rad6B. It binds to the Rad6B catalytic site, inhibits Rad6B-induced histone H2A ubiquitination, downregulates intracellular beta-catenin. It can induce G2/M arrest and apoptosis, and inhibit proliferation and migration of metastatic human breast cancer cells (IC50 ~6 µM).
Puffer: Powder
CAS Nummer: [1002789-86-7]