Exatecan Mesylate, CAS [[169869-90-3]]

Artikelnummer: BYT-ORB1296213
Artikelname: Exatecan Mesylate, CAS [[169869-90-3]]
Artikelnummer: BYT-ORB1296213
Hersteller Artikelnummer: orb1296213
Alternativnummer: BYT-ORB1296213-10, BYT-ORB1296213-100, BYT-ORB1296213-25, BYT-ORB1296213-50, BYT-ORB1296213-500
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: DX8951f, ADC Cytotoxin, ADCCytotoxin, Exatecan, Exatecan Mesylate, Inhibitor, inhibit, Topoisomerase, Topo I
Exatecan Mesylate (DX-8951f) is a potent inhibitor of DNA topoisomerase I, exhibiting an IC50 of 2.2 µM. This camptothecin analog has demonstrated antitumor activity in both in vitro cytotoxicity assays and in vivo xenograft models, supporting its research use in oncology and cancer pharmacology.
Molekulargewicht: 531.55
Reinheit: 99.90% (May vary between batches)
CAS Nummer: [169869-90-3]
Formel: C25H26FN3O7S
Target-Kategorie: Topoisomerase,ADC Cytotoxin
Anwendungsbeschreibung: Solubility: H2O:6 mg/mL (11.29 mM),DMSO:8 mg/mL (15.05 mM)