Aticaprant, CAS [[1174130-61-0]]
Artikelnummer:
BYT-ORB1296218
Produktübersicht
Artikelname:
Aticaprant, CAS [[1174130-61-0]]
Artikelnummer:
BYT-ORB1296218
Hersteller Artikelnummer:
orb1296218
Alternativnummer:
BYT-ORB1296218-1, BYT-ORB1296218-1, BYT-ORB1296218-10, BYT-ORB1296218-100, BYT-ORB1296218-2, BYT-ORB1296218-25, BYT-ORB1296218-5, BYT-ORB1296218-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
CERC 501, CERC501, CERC-501, Aticaprant, Inhibitor, inhibit, Opioid Receptor, OpioidReceptor, LY 2456302, LY2456302, LY-2456302, kappa-opioid receptor
Produktbeschreibung
Aticaprant (CERC-501) is a highly potent and brain-penetrant kappa-opioid receptor (KOR) antagonist with a Ki of 0.807 nM. It is a valuable research tool for investigating KORs role in stress-related behaviors, depression, and addiction in both in vitro and in vivo preclinical models.
Produkteigenschaften
Molekulargewicht:
418.5
Reinheit:
99.97% (May vary between batches)
CAS Nummer:
[1174130-61-0]
Formel:
C26H27FN2O2
Target-Kategorie:
Opioid Receptor
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.56 mM),DMSO:100 mg/mL (238.95 mM)