Aticaprant, CAS [[1174130-61-0]]

Product Overview

• Article Name: Aticaprant, CAS [[1174130-61-0]]
• Biozol Catalog Number: BYT-ORB1296218
• Supplier Catalog Number: orb1296218
• Alternative Catalog Number: BYT-ORB1296218-1, BYT-ORB1296218-1, BYT-ORB1296218-10, BYT-ORB1296218-100, BYT-ORB1296218-2, BYT-ORB1296218-25, BYT-ORB1296218-5, BYT-ORB1296218-50
• Manufacturer: Biorbyt
• Category: Biochemikalien
• Alternative Names: CERC 501, CERC501, CERC-501, Aticaprant, Inhibitor, inhibit, Opioid Receptor, OpioidReceptor, LY 2456302, LY2456302, LY-2456302, kappa-opioid receptor

Product Description

Aticaprant (CERC-501) is a highly potent and brain-penetrant kappa-opioid receptor (KOR) antagonist with a Ki of 0.807 nM. It is a valuable research tool for investigating KORs role in stress-related behaviors, depression, and addiction in both in vitro and in vivo preclinical models.

Product Properties

• Molecular Weight: 418.5
• Purity: 99.97% (May vary between batches)
• CAS Number: [1174130-61-0]
• Formula: C26H27FN2O2
• Target: Opioid Receptor

Application Notes

• Application Notes: Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.56 mM),DMSO:100 mg/mL (238.95 mM)