Ningetinib Tosylate, CAS [[1394820-77-9]]
Artikelnummer:
BYT-ORB1296250
Produktübersicht
Artikelname:
Ningetinib Tosylate, CAS [[1394820-77-9]]
Artikelnummer:
BYT-ORB1296250
Hersteller Artikelnummer:
orb1296250
Alternativnummer:
BYT-ORB1296250-1, BYT-ORB1296250-10, BYT-ORB1296250-100, BYT-ORB1296250-25, BYT-ORB1296250-5, BYT-ORB1296250-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
cMet, c-Met, cMet/HGFR, c-Met/HGFR, AXL, Axl, HGFR, Mer, inhibit, Inhibitor, Ningetinib, Ningetinib Tosylate, TAM Receptor, TAMReceptor, Vascular endothelial growth factor receptor, VEGFR, VEGFR2, Tyro3
Produktbeschreibung
Ningetinib Tosylate is a potent, orally active small molecule inhibitor targeting Axl, VEGFR2, and c-Met kinases with IC50 values below 10 nM. It is utilized in preclinical cancer research, particularly in studies involving tumor angiogenesis, metastasis, and resistance mechanisms in both cellular and animal models.
Produkteigenschaften
Molekulargewicht:
728.79
Reinheit:
99.93% (May vary between batches)
CAS Nummer:
[1394820-77-9]
Formel:
C38H37FN4O8S
Target-Kategorie:
c-Met/HGFR,VEGFR,TAM Receptor
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: DMSO:8 mg/mL (10.98 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (1.37 mM)