Ningetinib, CAS [[1394820-69-9]]

Artikelnummer: BYT-ORB1296265
Artikelname: Ningetinib, CAS [[1394820-69-9]]
Artikelnummer: BYT-ORB1296265
Hersteller Artikelnummer: orb1296265
Alternativnummer: BYT-ORB1296265-1, BYT-ORB1296265-10, BYT-ORB1296265-100, BYT-ORB1296265-2, BYT-ORB1296265-25, BYT-ORB1296265-5, BYT-ORB1296265-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: inhibit, Ningetinib, HGFR, Inhibitor, Mer, AXL, Axl, cMet, cMet/HGFR, c-Met, c-Met/HGFR, CT053, CT-053, CT053PTSA, CT 053, TAM Receptor, TAMReceptor, Tyro3, VEGFR2, VEGFR, Vascular endothelial growth factor receptor
Ningetinib (CT-053) is a potent, orally active small molecule inhibitor targeting Axl, VEGFR2, and c-Met kinases with low nanomolar IC50 values. It is utilized in preclinical cancer research, particularly in studies investigating tumor angiogenesis, metastasis, and resistance mechanisms in both cellular and animal models.
Molekulargewicht: 556.58
Reinheit: 99.98% (May vary between batches)
CAS Nummer: [1394820-69-9]
Formel: C31H29FN4O5
Target-Kategorie: VEGFR,TAM Receptor,c-Met/HGFR
Anwendungsbeschreibung: Solubility: DMSO:15 mg/mL (26.95 mM)