GSK778 hydrochloride is a potent and selective BD1 bromodomain inhibitor of BET proteins, demonstrating low nanomolar IC50 values. It mimics pan-BET inhibitor effects in cancer models, making it a valuable tool for epigenetic research in oncology, applicable in both cellular and in vivo studies of transcriptional regulation and tumor progression.
Molekulargewicht:
548.08
Reinheit:
98.35% (May vary between batches)
CAS Nummer:
[2863657-79-6]
Formel:
C30H34ClN5O3
Target-Kategorie:
Apoptosis,Epigenetic Reader Domain
Anwendungsbeschreibung:
Solubility: DMSO:50 mg/mL (91.23 mM)
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten