GSK778 hydrochloride, CAS [[2863657-79-6]]

Artikelnummer: BYT-ORB1297936
Artikelname: GSK778 hydrochloride, CAS [[2863657-79-6]]
Artikelnummer: BYT-ORB1297936
Hersteller Artikelnummer: orb1297936
Alternativnummer: BYT-ORB1297936-1, BYT-ORB1297936-1, BYT-ORB1297936-10, BYT-ORB1297936-100, BYT-ORB1297936-25, BYT-ORB1297936-5, BYT-ORB1297936-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: BET, EpigeneticReaderDomain, Epigenetic Reader Domain, GSK-778 Hydrochloride, GSK778 Hydrochloride, GSK778 hydrochloride, GSK 778 Hydrochloride
GSK778 hydrochloride is a potent and selective BD1 bromodomain inhibitor of BET proteins, demonstrating low nanomolar IC50 values. It mimics pan-BET inhibitor effects in cancer models, making it a valuable tool for epigenetic research in oncology, applicable in both cellular and in vivo studies of transcriptional regulation and tumor progression.
Molekulargewicht: 548.08
Reinheit: 98.35% (May vary between batches)
CAS Nummer: [2863657-79-6]
Formel: C30H34ClN5O3
Target-Kategorie: Apoptosis,Epigenetic Reader Domain
Anwendungsbeschreibung: Solubility: DMSO:50 mg/mL (91.23 mM)