SHR0302, CAS [[1445987-21-2]]

Artikelnummer: BYT-ORB1298293
Artikelname: SHR0302, CAS [[1445987-21-2]]
Artikelnummer: BYT-ORB1298293
Hersteller Artikelnummer: orb1298293
Alternativnummer: BYT-ORB1298293-1, BYT-ORB1298293-1, BYT-ORB1298293-10, BYT-ORB1298293-100, BYT-ORB1298293-25, BYT-ORB1298293-5, BYT-ORB1298293-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: collagen, B-cell, arthritis, ARQ252, ARQ-252, ARQ 252, anti-inflammatory, anti-proliferation, Apoptosis, Inhibitor, Janus kinase, JAK1, JAK1-STAT3, JAK, inhibit, migration, fibrosis, hepatic, SHR 0302, SHR0302, SHR-0302, phosphorylation, Th17
SHR0302 (ARQ252) is a selective JAK1 inhibitor, demonstrating >10-fold selectivity over JAK2, 77-fold over JAK3, and 420-fold over Tyk2. This small molecule is a valuable research tool for investigating JAK1-dependent pathways in both cellular and animal models of autoimmune and inflammatory diseases.
Molekulargewicht: 414.48
Reinheit: 99.11% (May vary between batches)
CAS Nummer: [1445987-21-2]
Formel: C18H22N8O2S
Target-Kategorie: Apoptosis,JAK
Anwendungsbeschreibung: Solubility: 10% DMSO+40% PEG300+5% Tween-80+45% Saline:2 mg/mL (4.83 mM),DMSO:30 mg/mL (72.38 mM)