DS-1205, CAS [[1855860-24-0]]

Artikelnummer: BYT-ORB1298349
Artikelname: DS-1205, CAS [[1855860-24-0]]
Artikelnummer: BYT-ORB1298349
Hersteller Artikelnummer: orb1298349
Alternativnummer: BYT-ORB1298349-1, BYT-ORB1298349-1, BYT-ORB1298349-10, BYT-ORB1298349-25, BYT-ORB1298349-5
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: c-Met/HGFR, DS 1205, DS1205, DS-1205, DS-1205b, AXL, Axl, Inhibitor, Mer, NIH3T3, MET, migration, kinase, inhibit, Tropomyosin related kinase receptor, TRKA, Trk Receptor, Tyro3, tumor, TAM Receptor, TAMReceptor
DS-1205 is a highly potent and selective AXL kinase inhibitor (IC50 = 1.3 nM), with additional activity against MER, MET, and TRKA kinases. This small molecule has demonstrated efficacy in suppressing cell migration in vitro and impeding tumor growth in animal models, supporting its research use in oncology and metastasis studies.
Molekulargewicht: 735.8
Reinheit: 99.75% (May vary between batches)
CAS Nummer: [1855860-24-0]
Formel: C41H42FN5O7
Target-Kategorie: TAM Receptor,Trk receptor,c-Met/HGFR
Anwendungsbeschreibung: Solubility: DMSO:45 mg/mL (61.16 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (2.72 mM)