BMS-911543, CAS [[1271022-90-2]]
Artikelnummer:
BYT-ORB1300463
Produktübersicht
Artikelname:
BMS-911543, CAS [[1271022-90-2]]
Artikelnummer:
BYT-ORB1300463
Hersteller Artikelnummer:
orb1300463
Alternativnummer:
BYT-ORB1300463-1, BYT-ORB1300463-1, BYT-ORB1300463-5, BYT-ORB1300463-10, BYT-ORB1300463-25, BYT-ORB1300463-50
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
SET-2, Tyrosine Kinases, TyrosineKinases, TYK2, BMS 911543, BMS911543, BMS-911543, Inhibitor, HistoneMethyltransferase, Histone Methyltransferase, JAK3, Janus kinase, JAK2, JAK, JAK1, inhibit
Produktbeschreibung
BMS-911543 is a highly selective JAK2 inhibitor (IC50 = 1.1 nM) with significant selectivity over JAK1, JAK3, and TYK2. It is a valuable research tool for investigating JAK2-dependent pathways in myeloproliferative neoplasms and hematological malignancies, as evidenced in both in vitro and in vivo preclinical studies.
Produkteigenschaften
Molekulargewicht:
432.52
Reinheit:
99.98% (May vary between batches)
CAS Nummer:
[1271022-90-2]
Formel:
C23H28N8O
Target-Kategorie:
Histone Methyltransferase,Tyrosine Kinases,JAK
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (4.62 mM),DMSO:34 mg/mL (78.61 mM),H2O:< 1 mg/mL (insoluble or slightly soluble),Ethanol:21 mg/mL (48.55 mM)