Thioperamide maleate (MR-12842 maleate) is a potent and selective histamine H3 receptor antagonist, with a Ki of 4.3 nM for receptor binding and 31 nM for inhibiting [H]histamine synthesis. This compound is widely used in neuroscience research to study H3 receptor function in both in vitro and in vivo models of sleep, cognition, and energy homeostasis.
Molekulargewicht:
408.52
Reinheit:
99.88% (May vary between batches)
CAS Nummer:
[148440-81-7]
Formel:
C19H28N4O4S
Target-Kategorie:
Histamine Receptor
Anwendungsbeschreibung:
Solubility: DMSO:55 mg/mL (134.63 mM)
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten