PG01 is a potent CFTR chloride channel potentiator effective against multiple CFTR mutants, including deltaF508, E193K, G970R, and G551D, with sub-micromolar affinity. It corrects gating defects by enhancing forskolin-stimulated chloride currents, making it a valuable research tool for in vitro cystic fibrosis studies and CFTR pharmacology investigations.
Molekulargewicht:
439.55
Reinheit:
99.87% (May vary between batches)
CAS Nummer:
[853138-65-5]
Formel:
C28H29N3O2
Target-Kategorie:
CFTR
Anwendungsbeschreibung:
Solubility: DMSO:30 mg/mL (68.25 mM)
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten