AMG-009 is a potent small molecule dual antagonist targeting both the CRTH2 and DP receptors with high selectivity, exhibiting IC50 values of 3 nM and 12 nM, respectively. It is a valuable research tool for investigating the roles of these prostanoid receptors in allergic inflammation and asthma, applicable in both in vitro binding assays and in vivo disease models.
Molekulargewicht:
581.47
Reinheit:
97.88% (May vary between batches)
CAS Nummer:
[1027847-67-1]
Formel:
C26H26Cl2N2O7S
Target-Kategorie:
GPCR,Prostaglandin Receptor
Anwendungsbeschreibung:
Solubility: DMSO:100 mg/mL (171.98 mM)
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten