Neratinib maleate, CAS [[915942-22-2]]

Artikelnummer: BYT-ORB1944868
Artikelname: Neratinib maleate, CAS [[915942-22-2]]
Artikelnummer: BYT-ORB1944868
Hersteller Artikelnummer: orb1944868
Alternativnummer: BYT-ORB1944868-100, BYT-ORB1944868-25, BYT-ORB1944868-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: Neratinib Maleate, HKI 272 Maleate, HKI272 Maleate, HKI-272 Maleate, HKI-272 maleate, HER2, EGFR
Neratinib maleate is an irreversible, orally bioavailable inhibitor selectively targeting HER2 (IC50=59 nM) and EGFR (IC50=92 nM). It is widely used in preclinical cancer research, demonstrating antitumor activity in both in vitro assays and in vivo models for breast, prostate, and other solid tumors.
Molekulargewicht: 673.11
Reinheit: 99.99% (May vary between batches)
CAS Nummer: [915942-22-2]
Formel: C34H33ClN6O7
Target-Kategorie: HER,EGFR
Anwendungsbeschreibung: Solubility: DMSO:225 mg/mL (334.27 mM)