TM2 TEAD inhibitor, CAS [[1008768-41-9]]

Produktübersicht

• Artikelname: TM2 TEAD inhibitor, CAS [[1008768-41-9]]
• Artikelnummer: BYT-ORB1979922
• Hersteller Artikelnummer: orb1979922
• Alternativnummer: BYT-ORB1979922-1, BYT-ORB1979922-10, BYT-ORB1979922-100, BYT-ORB1979922-25, BYT-ORB1979922-5, BYT-ORB1979922-50
• Hersteller: Biorbyt
• Kategorie: Biochemikalien
• Alternative Synonym: TEAD-IN-8

Produktbeschreibung

TM2 is a potent, reversible TEAD inhibitor that blocks auto-palmitoylation (IC50: 38 nM TEAD4) and disrupts TEAD-YAP transcriptional activity. It demonstrates significant antiproliferative effects in YAP-dependent cancer cells and potently inhibits the growth of YAP-driven liver organoids in vitro, supporting its investigation as an anticancer therapeutic.

Produkteigenschaften

• Molekulargewicht: 435.57
• Reinheit: 99.91% (May vary between batches)
• CAS Nummer: [1008768-41-9]
• Formel: C26H33N3O3
• Target-Kategorie: YAP