Cell permeable, ATP-competitive inhibitor of the four isoforms of ribosomal S6 kinase (p90 RSK) (IC50s at 100µM ATP: RSK1 = 31nM, RSK2 = 24nM, RSK3 = 18nM, RSK4 = 15nM). Does not significantly inhibit 10 other AGC kinases, and over 40 other protein kinas
Molekulargewicht:
391.4
Reinheit:
98% (HPLC)
CAS Nummer:
[501437-28-1]
Formel:
C19H23F2N5O2
Target-Kategorie:
S6 kinase
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten