Cell permeable, ATP-competitive inhibitor of the four isoforms of ribosomal S6 kinase (p90 RSK) (IC50s at 100µM ATP: RSK1 = 31nM, RSK2 = 24nM, RSK3 = 18nM, RSK4 = 15nM). Does not significantly inhibit 10 other AGC kinases, and over 40 other protein kinas
Molecular Weight:
391.4
Purity:
98% (HPLC)
CAS Number:
[501437-28-1]
Formula:
C19H23F2N5O2
Target:
S6 kinase
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