Nelfinavir mesylate, CAS [[159989-65-8]]

Artikelnummer: FBM-10-3050
Artikelname: Nelfinavir mesylate, CAS [[159989-65-8]]
Artikelnummer: FBM-10-3050
Hersteller Artikelnummer: 10-3050
Alternativnummer: FBM-10-3050-10MG,FBM-10-3050-50MG
Hersteller: Focus Biomolecules
Kategorie: Biochemikalien
Alternative Synonym: AG-1343
HIV Protease inhibitor / Anticancer activity
Molekulargewicht: 663.88
Reinheit: 98% by HPLC NMR (conforms)
Formulierung: White solid
CAS Nummer: [159989-65-8]
Formel: C32H45N3O4S CH3SO3H
Anwendungsbeschreibung: Nelfinavir is a clinically useful anti-HIV agent acting via inhibition of HIV-1 protease (Ki=2 nM).1 It also displays efficacy in cancer, malaria, tuberculosis and SARS.2 Displays broad spectrum anticancer activity and induces endoplasmic reticulum stress, autophagy and apoptosis in vitro and in vivo.3 Inhibits the growth of HER2-positive breast cancer cells via inhibition of HSP90 through a novel mechanism.4