Nevanimibe hydrochloride, CAS [[133825-81-7]]

Artikelnummer: MCE-HY-100399A
Artikelname: Nevanimibe hydrochloride, CAS [[133825-81-7]]
Artikelnummer: MCE-HY-100399A
Hersteller Artikelnummer: HY-100399A
Alternativnummer: MCE-HY-100399A-10MG,MCE-HY-100399A-50MG,MCE-HY-100399A-10MMX1ML,MCE-HY-100399A-100MG,MCE-HY-100399A-5MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: PD-132301 hydrochloride, ATR101 hydrochloride
Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) inhibitor with an EC50 of 9 nM. Nevanimibe hydrochloride inhibits ACAT2 with an EC50 of 368 nM. Nevanimibe hydrochloride induces cell apoptosis and has the potential for adrenocortical cancer[1].
Molekulargewicht: 458.08
Reinheit: 99.49
CAS Nummer: [133825-81-7]
Formel: C27H40ClN3O
Target-Kategorie: Acyltransferase,Apoptosis
Anwendungsbeschreibung: Reference compound