CPI-455 (hydrochloride), CAS [[2095432-28-1]]

Artikelnummer: MCE-HY-100421A
Artikelname: CPI-455 (hydrochloride), CAS [[2095432-28-1]]
Artikelnummer: MCE-HY-100421A
Hersteller Artikelnummer: HY-100421A
Alternativnummer: MCE-HY-100421A-10MG,MCE-HY-100421A-5MG,MCE-HY-100421A-1MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
CPI-455 hydrochloride is a specific, pan-KDM5 inhibitor with an IC50 of 10 nM for KDM5A. CPI-455 hydrochloride mediates KDM5 inhibition, elevates global levels of H3K4me3, and decreases the number of drug-tolerant persister cancer cells in multiple cancer cell line models treated with standard chemotherapy or targeted agents[1].
Molekulargewicht: 314.77
Reinheit: 99.95
CAS Nummer: [2095432-28-1]
Formel: C16H15ClN4O
Target-Kategorie: Histone Demethylase
Anwendungsbeschreibung: Reference compound