TAK-243, CAS [[1450833-55-2]]

Artikelnummer: MCE-HY-100487
Artikelname: TAK-243, CAS [[1450833-55-2]]
Artikelnummer: MCE-HY-100487
Hersteller Artikelnummer: HY-100487
Alternativnummer: MCE-HY-100487-50MG,MCE-HY-100487-10MG,MCE-HY-100487-10MMX1ML,MCE-HY-100487-100MG,MCE-HY-100487-5MG,MCE-HY-100487-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: MLN7243
TAK-243 (MLN7243) is a first-in-class, selective ubiquitin activating enzyme, UAE (UBA1) inhibitor (IC50=1 nM), which blocks ubiquitin conjugation, disrupting monoubiquitin signaling as well as global protein ubiquitination. TAK-243 (MLN7243) induces endoplasmic reticulum (ER) stress, abrogates NF-kappaB pathway activation and promotes apoptosis[1][2].
Molekulargewicht: 519.52
Reinheit: 98.38
CAS Nummer: [1450833-55-2]
Formel: C19H20F3N5O5S2
Target-Kategorie: Apoptosis,E1/E2/E3 Enzyme,NF-kappaB
Anwendungsbeschreibung: MCE Product type: Reference compound