Lesogaberan (hydrochloride) (Standard), CAS [[2925644-17-1]] Preis auf Anfrage
Artikelnummer:
MCE-HY-10061BR
Hersteller Artikelnummer:
HY-10061BR
Alternativnummer:
MCE-HY-10061BR-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Lesogaberan (hydrochloride) (Standard) is the analytical standard of Lesogaberan (hydrochloride) (HY-10061B). This product is intended for research and analytical applications. Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptor. The affinity (Kis) of Lesogaberan hydrochloride for rat GABAB and GABAA receptors, as measured by displacement of [3H]GABA binding in brain membranes: 5.1 nM and 1.4 µM, respectively. Lesogaberan hydrochloride inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action[1].
Molekulargewicht:
177.54
CAS Nummer:
[2925644-17-1]
Formel:
C3H10ClFNO2P
Target-Kategorie:
GABA Receptor,Reference Standards
Anwendungsbeschreibung:
MCE Product type: Reference Standards
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten