Lesogaberan (hydrochloride) (Standard), CAS [[2925644-17-1]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-10061BR
Supplier Catalog Number:
HY-10061BR
Alternative Catalog Number:
MCE-HY-10061BR-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Lesogaberan (hydrochloride) (Standard) is the analytical standard of Lesogaberan (hydrochloride) (HY-10061B). This product is intended for research and analytical applications. Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptor. The affinity (Kis) of Lesogaberan hydrochloride for rat GABAB and GABAA receptors, as measured by displacement of [3H]GABA binding in brain membranes: 5.1 nM and 1.4 µM, respectively. Lesogaberan hydrochloride inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action[1].
Molecular Weight:
177.54
CAS Number:
[2925644-17-1]
Formula:
C3H10ClFNO2P
Target:
GABA Receptor,Reference Standards
Application Notes:
MCE Product type: Reference Standards
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