FG 7142, CAS [[78538-74-6]]

Artikelnummer: MCE-HY-100991
Artikelname: FG 7142, CAS [[78538-74-6]]
Artikelnummer: MCE-HY-100991
Hersteller Artikelnummer: HY-100991
Alternativnummer: MCE-HY-100991-2MG,MCE-HY-100991-25MG,MCE-HY-100991-10MMX1ML,MCE-HY-100991-5MG,MCE-HY-100991-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: ZK 39106, LSU-65
FG 7142 (ZK 39106, LSU-65), a non-selectively benzodiazepine inverse agonist, has high affinity for the alpha1 subunit-containing GABAA receptor (Ki=91 nM). FG 7142 (ZK 39106, LSU-65) also modulates GABA-induced chloride flux at GABAA receptors expressing the alpha1 subunit (EC50= 137 nM). FG 7142 (ZK 39106, LSU-65) can increase tyrosine hydroxylation and cause upregulation of beta-adrenoceptors in mouse cerebral cortex[1].
Molekulargewicht: 225.25
Reinheit: 99.43
CAS Nummer: [78538-74-6]
Formel: C13H11N3O
Target-Kategorie: GABA Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound1