Relacatib, CAS [[362505-84-8]]

Produktübersicht

• Artikelname: Relacatib, CAS [[362505-84-8]]
• Artikelnummer: MCE-HY-10294
• Hersteller Artikelnummer: HY-10294
• Alternativnummer: MCE-HY-10294-1MG,MCE-HY-10294-25MG,MCE-HY-10294-5MG,MCE-HY-10294-10MMX1ML,MCE-HY-10294-10MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: SB-462795

Produktbeschreibung

Relacatib (SB-462795) is a novel, potent, and orally active inhibitor of human cathepsins K, L, and V with Ki values of 41 pM, 68 pM, and 53 pM, respectively. Relacatib inhibits endogenous cathepsin K in situ in human osteoclasts and human osteoclast-mediated bone resorption with IC50 values of 45 nM and 70 nM, respectively. Relacatib inhibits bone resorption in vitro in human tissue as well as in cynomolgus monkeys in vivo[1][2].

Produkteigenschaften

• Molekulargewicht: 540.63
• Reinheit: 99.99
• CAS Nummer: [362505-84-8]
• Formel: C27H32N4O6S
• Target-Kategorie: Cathepsin

Anwendungsbeschreibung

• Anwendungsbeschreibung: Reference compound