Relacatib, CAS [[362505-84-8]]

Product Overview

• Article Name: Relacatib, CAS [[362505-84-8]]
• Biozol Catalog Number: MCE-HY-10294
• Supplier Catalog Number: HY-10294
• Alternative Catalog Number: MCE-HY-10294-1MG,MCE-HY-10294-25MG,MCE-HY-10294-5MG,MCE-HY-10294-10MMX1ML,MCE-HY-10294-10MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: SB-462795

Product Description

Relacatib (SB-462795) is a novel, potent, and orally active inhibitor of human cathepsins K, L, and V with Ki values of 41 pM, 68 pM, and 53 pM, respectively. Relacatib inhibits endogenous cathepsin K in situ in human osteoclasts and human osteoclast-mediated bone resorption with IC50 values of 45 nM and 70 nM, respectively. Relacatib inhibits bone resorption in vitro in human tissue as well as in cynomolgus monkeys in vivo[1][2].

Product Properties

• Molecular Weight: 540.63
• Purity: 99.99
• CAS Number: [362505-84-8]
• Formula: C27H32N4O6S
• Target: Cathepsin

Application Notes

• Application Notes: Reference compound