Relacatib (Standard), CAS [[362505-84-8]] Preis auf Anfrage

Produktübersicht

• Artikelname: Relacatib (Standard), CAS [[362505-84-8]] Preis auf Anfrage
• Artikelnummer: MCE-HY-10294R
• Hersteller Artikelnummer: HY-10294R
• Alternativnummer: MCE-HY-10294R-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

Relacatib (Standard) is the analytical standard of Relacatib (HY-10294). This product is intended for research and analytical applications. Relacatib (SB-462795) is a novel, potent, and orally active inhibitor of human cathepsins K, L, and V with Ki values of 41 pM, 68 pM, and 53 pM, respectively. Relacatib inhibits endogenous cathepsin K in situ in human osteoclasts and human osteoclast-mediated bone resorption with IC50 values of 45 nM and 70 nM, respectively. Relacatib inhibits bone resorption in vitro in human tissue as well as in cynomolgus monkeys in vivo[1][2].

Produkteigenschaften

• Molekulargewicht: 540.63
• CAS Nummer: [362505-84-8]
• Formel: C27H32N4O6S
• Target-Kategorie: Cathepsin,Reference Standards

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference Standards