Relacatib (Standard), CAS [[362505-84-8]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-10294R
Supplier Catalog Number:
HY-10294R
Alternative Catalog Number:
MCE-HY-10294R-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Relacatib (Standard) is the analytical standard of Relacatib (HY-10294). This product is intended for research and analytical applications. Relacatib (SB-462795) is a novel, potent, and orally active inhibitor of human cathepsins K, L, and V with Ki values of 41 pM, 68 pM, and 53 pM, respectively. Relacatib inhibits endogenous cathepsin K in situ in human osteoclasts and human osteoclast-mediated bone resorption with IC50 values of 45 nM and 70 nM, respectively. Relacatib inhibits bone resorption in vitro in human tissue as well as in cynomolgus monkeys in vivo[1][2].
Molecular Weight:
540.63
CAS Number:
[362505-84-8]
Formula:
C27H32N4O6S
Target:
Cathepsin,Reference Standards
Application Notes:
MCE Product type: Reference Standards
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