(S)-SNAP5114, CAS [[157604-55-2]]

Produktübersicht

• Artikelname: (S)-SNAP5114, CAS [[157604-55-2]]
• Artikelnummer: MCE-HY-103504
• Hersteller Artikelnummer: HY-103504
• Alternativnummer: MCE-HY-103504-25MG,MCE-HY-103504-50MG,MCE-HY-103504-100MG,MCE-HY-103504-10MG,MCE-HY-103504-10MMX1ML,MCE-HY-103504-5MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

(S)-SNAP5114 is a non-covalent murine GABA transporter inhibitor with blood-brain barrier penetration ability, which exhibits significant subtype-selective inhibitory activity against mGAT4 (pIC50=5.71, pKi=4.56), much higher than its effects on mGAT1, mGAT2 and mGAT3. (S)-SNAP5114 elevates extracellular GABA concentrations by blocking the GABA reuptake mechanism, thereby enhancing thalamus-specific GABAergic signaling and exerting potential neuromodulatory effects. (S)-SNAP5114 is widely used in studies related to epilepsy, neuropathic pain, anxiety and depression, and various neurodegenerative diseases[1][2][3].

Produkteigenschaften

• Molekulargewicht: 505.60
• Reinheit: 98.09
• CAS Nummer: [157604-55-2]
• Formel: C30H35NO6
• Target-Kategorie: GABA Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound1