Upidosin (Rec 15/2739) is an alpha-1 adrenoceptor (alpha-1 AR) antagonist. Upidosin shows moderate selectivity for the alpha-1A AR subtype. Upidosin shows uroselectivity in urethra and prostate with a Kb value of 2-3 nM higher than in ear artery and aorta with a Kb value of 20-100 nM. Upidosin inhibits [3H]prazosin binding to cloned human alpha-1A adrenergic receptor. Upidosin can be used for the research of urethral obstruction[1].
Molekulargewicht:
511.61
Reinheit:
99.48
CAS Nummer:
[152735-23-4]
Formel:
C31H33N3O4
Target-Kategorie:
Adrenergic Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten