Upidosin (Rec 15/2739) is an alpha-1 adrenoceptor (alpha-1 AR) antagonist. Upidosin shows moderate selectivity for the alpha-1A AR subtype. Upidosin shows uroselectivity in urethra and prostate with a Kb value of 2-3 nM higher than in ear artery and aorta with a Kb value of 20-100 nM. Upidosin inhibits [3H]prazosin binding to cloned human alpha-1A adrenergic receptor. Upidosin can be used for the research of urethral obstruction[1].
Molecular Weight:
511.61
Purity:
99.48
CAS Number:
[152735-23-4]
Formula:
C31H33N3O4
Target:
Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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