5-Guanidinonaltrindole (TFA), CAS [[219655-57-9]] Preis auf Anfrage

Produktübersicht

• Artikelname: 5-Guanidinonaltrindole (TFA), CAS [[219655-57-9]] Preis auf Anfrage
• Artikelnummer: MCE-HY-107748A
• Hersteller Artikelnummer: HY-107748A
• Alternativnummer: MCE-HY-107748A-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: 5-GNTI (TFA)

Produktbeschreibung

5-Guanidinonaltrindole TFA is a selective kappa-opioid receptor antagonist with significant opioid antagonist activity. 5-Guanidinonaltrindole TFA exhibits 5 times the antagonistic potency of the prototypical kappa-opioid receptor antagonist norbinatorphimine in smooth muscle preparations, with a selectivity ratio exceeding 500 times. Binding and functional studies of 5-Guanidinonaltrindole TFA showed pA(2) values comparable to smooth muscle data. 5-Guanidinonaltrindole TFA is regarded as a potentially valuable pharmacological tool for studying opioids due to its high selectivity and potency[1].

Produkteigenschaften

• Molekulargewicht: 699.60
• CAS Nummer: [219655-57-9]
• Formel: C31H31F6N5O7
• Target-Kategorie: Endogenous Metabolite

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound