5-Guanidinonaltrindole (TFA), CAS [[219655-57-9]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-107748A
Supplier Catalog Number:
HY-107748A
Alternative Catalog Number:
MCE-HY-107748A-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
5-GNTI (TFA)
5-Guanidinonaltrindole TFA is a selective kappa-opioid receptor antagonist with significant opioid antagonist activity. 5-Guanidinonaltrindole TFA exhibits 5 times the antagonistic potency of the prototypical kappa-opioid receptor antagonist norbinatorphimine in smooth muscle preparations, with a selectivity ratio exceeding 500 times. Binding and functional studies of 5-Guanidinonaltrindole TFA showed pA(2) values comparable to smooth muscle data. 5-Guanidinonaltrindole TFA is regarded as a potentially valuable pharmacological tool for studying opioids due to its high selectivity and potency[1].
Molecular Weight:
699.60
CAS Number:
[219655-57-9]
Formula:
C31H31F6N5O7
Target:
Endogenous Metabolite
Application Notes:
MCE Product type: Reference compound
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