CP-100356 (hydrochloride), CAS [[142715-48-8]]

Produktübersicht

• Artikelname: CP-100356 (hydrochloride), CAS [[142715-48-8]]
• Artikelnummer: MCE-HY-108347
• Hersteller Artikelnummer: HY-108347
• Alternativnummer: MCE-HY-108347-5MG,MCE-HY-108347-50MG,MCE-HY-108347-10MG,MCE-HY-108347-25MG,MCE-HY-108347-100MG,MCE-HY-108347-10MMX1ML
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

CP-100356 hydrochloride is an orally active dual MDR1 (P-gp)/BCRP inhibitor, with an IC50s of 0.5 and 1.5 µM for inhibiting MDR1-mediated Calcein-AM transport and BCRP-mediated Prazosin transport, respectively. CP-100356 hydrochloride is also a weak inhibitor of OATP1B1 (IC50=66 µM). CP-100356 hydrochloride is devoid of inhibition against MRP2 and major human P450 enzymes (IC50>15 µM)[1].

Produkteigenschaften

• Molekulargewicht: 597.10
• Reinheit: 99.68
• CAS Nummer: [142715-48-8]
• Formel: C31H37ClN4O6
• Target-Kategorie: BCRP,P-glycoprotein

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound