CP-100356 (hydrochloride), CAS [[142715-48-8]]

Product Overview

• Article Name: CP-100356 (hydrochloride), CAS [[142715-48-8]]
• Biozol Catalog Number: MCE-HY-108347
• Supplier Catalog Number: HY-108347
• Alternative Catalog Number: MCE-HY-108347-25MG,MCE-HY-108347-100MG,MCE-HY-108347-50MG,MCE-HY-108347-10MG,MCE-HY-108347-10MMX1ML,MCE-HY-108347-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

CP-100356 hydrochloride is an orally active dual MDR1 (P-gp)/BCRP inhibitor, with an IC50s of 0.5 and 1.5 µM for inhibiting MDR1-mediated Calcein-AM transport and BCRP-mediated Prazosin transport, respectively. CP-100356 hydrochloride is also a weak inhibitor of OATP1B1 (IC50=66 µM). CP-100356 hydrochloride is devoid of inhibition against MRP2 and major human P450 enzymes (IC50>15 µM)[1].

Product Properties

• Molecular Weight: 597.10
• Purity: 99.68
• CAS Number: [142715-48-8]
• Formula: C31H37ClN4O6
• Target: BCRP,P-glycoprotein

Application Notes

• Application Notes: Reference compound