GNE-781, CAS [[1936422-33-1]]

Produktübersicht

• Artikelname: GNE-781, CAS [[1936422-33-1]]
• Artikelnummer: MCE-HY-108696
• Hersteller Artikelnummer: HY-108696
• Alternativnummer: MCE-HY-108696-50MG,MCE-HY-108696-5MG,MCE-HY-108696-10MG,MCE-HY-108696-100MG,MCE-HY-108696-25MG,MCE-HY-108696-1MG,MCE-HY-108696-10MMX1ML
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

GNE-781 is an orally active, highly potent and selective CBP inhibitor with an IC50 of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET and BRD4(1) with IC50s of 6.2 nM and 5100 nM, respectively. GNE-781 displays antitumor activity in an MOLM-16 AML xenograft model[1].

Produkteigenschaften

• Molekulargewicht: 525.59
• Reinheit: 98.16
• CAS Nummer: [1936422-33-1]
• Formel: C27H33F2N7O2
• Target-Kategorie: Epigenetic Reader Domain,Histone Acetyltransferase

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound