Irdabisant (hydrochloride), CAS [[1005398-61-7]] Preis auf Anfrage

Produktübersicht

• Artikelname: Irdabisant (hydrochloride), CAS [[1005398-61-7]] Preis auf Anfrage
• Artikelnummer: MCE-HY-109968A
• Hersteller Artikelnummer: HY-109968A
• Alternativnummer: MCE-HY-109968A-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: CEP-26401 (hydrochloride)

Produktbeschreibung

Irdabisant (CEP-26401) hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist with Ki values of 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively. Irdabisant hydrochloride has relatively low inhibitory activity against hERG current with an IC50 of 13.8 µM. Irdabisant hydrochloride has cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant hydrochloride can be used to research schizophrenia or cognitive impairment[1][2].

Produkteigenschaften

• Molekulargewicht: 349.86
• CAS Nummer: [1005398-61-7]
• Formel: C18H24ClN3O2
• Target-Kategorie: Histamine Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound