Irdabisant (hydrochloride), CAS [[1005398-61-7]] Preis auf Anfrage

Product Overview

• Article Name: Irdabisant (hydrochloride), CAS [[1005398-61-7]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-109968A
• Supplier Catalog Number: HY-109968A
• Alternative Catalog Number: MCE-HY-109968A-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: CEP-26401 (hydrochloride)

Product Description

Irdabisant (CEP-26401) hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist with Ki values of 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively. Irdabisant hydrochloride has relatively low inhibitory activity against hERG current with an IC50 of 13.8 µM. Irdabisant hydrochloride has cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant hydrochloride can be used to research schizophrenia or cognitive impairment[1][2].

Product Properties

• Molecular Weight: 349.86
• CAS Number: [1005398-61-7]
• Formula: C18H24ClN3O2
• Target: Histamine Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound