(S)-PFI-2 (hydrochloride), CAS [[1627607-88-8]] Preis auf Anfrage

Produktübersicht

• Artikelname: (S)-PFI-2 (hydrochloride), CAS [[1627607-88-8]] Preis auf Anfrage
• Artikelnummer: MCE-HY-110196
• Hersteller Artikelnummer: HY-110196
• Alternativnummer: MCE-HY-110196-5MG,MCE-HY-110196-1MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

(S)-PFI-2 hydrochloride is an inhibitor of lysine methyltransferase SETD7 and is approximately 500-fold more active than its enantiomer (R)-PFI-2. (R)-PFI-2 is a cofactor-dependent and substrate-competitive inhibitor. (R)-PFI-2 can occupy the substrate peptide binding groove of SETD7 (including the catalytic lysine binding channel) and interact with the cofactor The donor methyl group is in direct contact. However, (S)-PFI-2 was not observed to have the same interaction as (R)-PFI-2[1][2].

Produkteigenschaften

• Molekulargewicht: 535.98
• CAS Nummer: [1627607-88-8]
• Formel: C23H26ClF4N3O3S
• Target-Kategorie: Histone Methyltransferase

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound