PHA-665752, CAS [[477575-56-7]]

Artikelnummer: MCE-HY-11107
Artikelname: PHA-665752, CAS [[477575-56-7]]
Artikelnummer: MCE-HY-11107
Hersteller Artikelnummer: HY-11107
Alternativnummer: MCE-HY-11107-10MG,MCE-HY-11107-5MG,MCE-HY-11107-10MMX1ML,MCE-HY-11107-25MG,MCE-HY-11107-50MG,MCE-HY-11107-100MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PHA-665752 is a selective, ATP-competitive, and active-site inhibitor of the catalytic activity of c-Met kinase (Ki=4 nM, IC50=9 nM). PHA-665752 exhibits >50-fold selectivity for c-Met compared with a panel of diverse tyrosine and serine-threonine kinases. PHA-665752 induces apoptosis and cell cycle arrest, and exhibits cytoreductive antitumor activity[1][2].
Molekulargewicht: 641.61
Reinheit: 98.74
CAS Nummer: [477575-56-7]
Formel: C32H34Cl2N4O4S
Target-Kategorie: Apoptosis,Autophagy,c-Met/HGFR
Anwendungsbeschreibung: MCE Product type: Reference compound