R406 (free base), CAS [[841290-80-0]]

Artikelnummer: MCE-HY-11108
Artikelname: R406 (free base), CAS [[841290-80-0]]
Artikelnummer: MCE-HY-11108
Hersteller Artikelnummer: HY-11108
Alternativnummer: MCE-HY-11108-5MG,MCE-HY-11108-10MG,MCE-HY-11108-50MG,MCE-HY-11108-100MG,MCE-HY-11108-1MG,MCE-HY-11108-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
R406 free base is an orally available and competitive Syk/FLT3 inhibitor for ATP binding with a Ki of 30 nM, potently inhibits Syk kinase activity in vitro with an IC50 of 41 nM, measured at an ATP concentration corresponding to its Km value. R406 free base reduces immune complex-mediated inflammation[1]. R406 free base also inhibits Lyn (IC50=63 nM) and Lck (IC50=37 nM)[2].
Molekulargewicht: 470.45
Reinheit: 99.07
CAS Nummer: [841290-80-0]
Formel: C22H23FN6O5
Target-Kategorie: Apoptosis,FLT3,Syk
Anwendungsbeschreibung: MCE Product type: Reference compound